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TOP 研究内容 メンバー 教室風景行事学会活動論文発表卒業後進路 工業的所有権 掲示板

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Publications (2007)



6 A Versatile Synthesis of a -Amino Acid Derivatives The Ugi Four-Component Condensation with a Novel Convertible sonitrile:
Kentaro Rikimaru, Arata Yanagisawa, Toshiyuki Kan, Tohru Fukuyama.
HETEROCYCLES, 73, 403-417,(2007) DOI: 10.3987/COM-07-S(U)11





5 Discrimination of carbonyl groups of meso--diketones with Horner -Wadsworth-Emmons reagent of chiral binaphthyl esters:
Daiki Monguchi, Yoshihisa Ohta, Tatsuya Yoshiuchi, Toshiyuki Watanabe, Takumi Furuta, Kiyoshi Tanaka and Kaoru Fuji
Tetrahedron, 63, 12712-12719 (2007). DOI: 10.1016/j.tet.2007.10.006




4 Divergent Synthesis of Multifunctional Molecular Probes Enabled Elucidation of the Enzyme Specificity of Dipeptidic γ-Secretase Inhibitors on Presenilin-Type Aspartic Proteases
Haruhiko Fuwa, Yasuko Takahashi, Yu Konno, Naoto Watanabe, Hiroyuki Miyashita, Makoto Sasaki, Hideaki Natsugari, Toshiyuki Kan, Tohru Fukuyama, Taisuke Tomita,Takeshi Iwatsubo.
ACS Chemical Biology2, 408-418 (2007)DOI: 10.1021/cb700073y





3 Convenient Synthesis of Photoaffinity Probes and Evaluation of Their Labeling Abilities:
Toshiyuki Kan, Yoichi Kita, Yuichi Morohashi, Yusuke Tominari, Shinnosuke Hosoda, Taisuke Tomita, Hideaki Natsugari, Takeshi Iwatsubo,Tohru Fukuyama.
Org. Lett., 9, 2055-2058 (2007).DOI: 10.1021/ol070376i





2 Concise synthesis of dideoxy-epigallocatechin gallate (DO-EGCG) and evaluation of its anti-influenza virus activity:
Takumi Furuta, Yasuo Hirooka, Ayako Abe, Yusuke Sugata, Mitsuru Ueda, Kouki Murakami, Takashi Suzuki, Kiyoshi Tanaka and Toshiyuki Kan
Bioorg. Med. Chem. Lett., 17, 3095-3098 (2007).DOI: 10.1016/j.bmcl.2007.03.041




1 Efficient synthesis of phenanthridinone derivatives via a palladium-catalyzed coupling process:
Takumi Furuta, Yuki Kitamura, Ayano Hashimoto, Satoshi Fujii, Kiyoshi Tanaka and Toshiyuki Kan.
Org. Lett., 9, 183-186 (2007)..DOI: 10.1021/ol062599z




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